Remove 2005 Remove Metabolic Stability Remove Research
article thumbnail

How the AI revolution can accelerate early drug discovery

Drug Target Review

Complex challenges such as metabolic stability or absorption, distribution, metabolism or excretion (ADME) properties could be better predicted, accurately filtering out poor candidates and streamlining discovery. Research and Development in the Pharmaceutical Industry | Congressional Budget Office [Internet].

Drugs 105
article thumbnail

Metabolism of five membered nitrogen containing heterocycles

Metabolite Tales Blog

Bicyclic structures containing five membered rings such as indoles, consisting of a six-membered benzene ring fused to a five-membered pyrrole ring, are also increasingly relevant as growing research fields such as psychedelics make use of these scaffolds, often found in natural products. 2009, 41, 157-167 [link] 19 Molecules.