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Game-changing pan-TEAD inhibitor for solid tumours

Drug Target Review

Leveraging AI-guided structure-based drug design, Insilico’s research and development team generated an impressive portfolio of over 6,000 molecules and identified three highly promising hit series. He is an adjunct professor of artificial intelligence at the Buck Institute for Research on Aging.

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Metabolism of five membered nitrogen containing heterocycles

Metabolite Tales Blog

Bicyclic structures containing five membered rings such as indoles, consisting of a six-membered benzene ring fused to a five-membered pyrrole ring, are also increasingly relevant as growing research fields such as psychedelics make use of these scaffolds, often found in natural products. 2006 , 34, 145-51 [link] 3 Drug Metab.