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Obstacles and innovations of macrocyclic drug development

Drug Target Review

Food and Drug Administration (FDA) approved drugs, macrocycles are used to combat a range of diseases, including cancer, viral, fungal and bacterial infections, neurodegenerative and autoimmune diseases. Nature Reviews Drug Discovery , 7(7):608624, 2008. 5 Macrocycles as drugs Despite accounting for just four percent of the U.S.