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Obstacles and innovations of macrocyclic drug development

Drug Target Review

Nature Reviews Drug Discovery , 7(7):608624, 2008. Cyclic Peptide Design, Chapter 2: Strategies to Enhance Metabolic Stabilities. Advanced Drug Delivery Reviews , 64:417, 2012. Driggers EM, Hale SP, Lee J, Terrett NK. The exploration of macrocycles for drug discovery: An underexploited structural class. Springer, 2019.