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Metabolism of five membered nitrogen containing heterocycles

Metabolite Tales Blog

2009, 41, 157-167 [link] 19 Molecules. 2010, 75, 9, 3141–3143 [link] 22 Clin Pharmacokinet. 44, 797–814 [link] Take a look at our other blogs The post Metabolism of five membered nitrogen containing heterocycles appeared first on Hypha Discovery. 2020, 25, 4309 [link] 20 Drug Metab. 2013, 41, 508-517 [link] 21 J.

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Efficient trajectories

Molecular Design

Design decisions in lead optimization are typically supported by assays for a range of properties such as solubility, permeability, metabolic stability and off-target activity as well as pharmacokinetic studies.