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Obstacles and innovations of macrocyclic drug development

Drug Target Review

Advanced Drug Delivery Reviews , 64:417, 2012. Cyclic Peptide Design, Chapter 2: Strategies to Enhance Metabolic Stabilities. References Lipinski CA, Lombardo F, Dominy BW, Feeney PJ. Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings. Springer, 2019.