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Obstacles and innovations of macrocyclic drug development

Drug Target Review

Nature Chemical Biology , 10(9):696698, 2014. Cyclic Peptide Design, Chapter 2: Strategies to Enhance Metabolic Stabilities. Macrocycles as protein-protein interaction inhibitors. Biochemical Journal , 474(7):11091125, 2017. Tools and rules for macrocycles. Jain AN, Brueckner AC, Jorge C, et al. Springer, 2019.