Metabolism of macrocyclic drugs
Metabolite Tales Blog
JULY 5, 2023
Journal of Medicinal Chemistry, 66 (8), 5377-5396. Journal of Medicinal Chemistry 62 (21), 9418-9437. link] [4] Macrocyclization via Ring-Closing Metathesis in Drug Discovery & Process Chemistry. Drug Hunter article, June 2023. References [1] Macrocycles in Drug Discovery─Learning from the Past for the Future.
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